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Search Results for " dna alkylation "

6

抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T11120 Duocarmycin TM

DNA Alkylation; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Duocarmycin TM 是一种有抗肿瘤活性的抗生素,也是一种 DNA 烷化剂。
T0923 Busulfan

Myleran,Sulphabutin,白消安,Busulphan

Apoptosis; DNA Alkylator/Crosslinker; DNA Alkylation Apoptosis; DNA Damage/DNA Repair
Busulfan (Busulphan) 是二甲磺酸盐的合成衍生物,具有抗肿瘤和细胞毒特性。是一种烷化剂,对骨髓具有选择性免疫抑制作用。
T1488 Procarbazine hydrochloride

NSC-77213 HCl,盐酸甲基苄肼,Procarbazine HCl

DNA Alkylator/Crosslinker; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Procarbazine hydrochloride (NSC-77213 HCl) 是一种烷化剂,是甲基肼衍生物的盐酸盐,具有抗肿瘤和诱变活性。
T31551 Mipicoledine

DMCHOCPEN,DM-CHOC-PEN,DM CHOC PEN

DM-CHOC-PEN is a DNA alkylation agent that may be used to treat brain cancer.
T11118 Duocarmycin SA

Others Others
Duocarmycin SA is an extremely potent cytotoxic agent and antitumor antibiotic that induces sequence-selective alkylation of duplex DNA, with an IC50 of 10 pM. It demonstrates synergistic cytotoxicity against glioblastoma multiforme (GBM) cells when combined with proton radiation in vitro.
T10973 DC41SMe

Others Others
DC41SMe is a DC1 derivative that is cytotoxic to Ramos, Namalwa and HL60 / s with IC50s ranging from 18-25 pM. DC1 is a simplified analogue of CC-1065, an antibody conjugate of cytotoxic DNA alkylation molecules, used for targeted treatment of cancer.

化合物

Duocarmycin TM
Cat.No: T11120
Synonym:
Target: DNA Alkylation, Antibiotic
Busulfan
Cat.No: T0923
Synonym: Myleran,Sulphabutin,白消安,Busulphan
Target: Apoptosis, DNA Alkylator/Crosslinker, DNA Alkylation
Procarbazine hydrochloride
Cat.No: T1488
Synonym: NSC-77213 HCl,盐酸甲基苄肼,Procarbazine HCl
Target: DNA Alkylator/Crosslinker, DNA/RNA Synthesis
Mipicoledine
Cat.No: T31551
Synonym: DMCHOCPEN,DM-CHOC-PEN,DM CHOC PEN
Target:
Duocarmycin SA
Cat.No: T11118
Synonym:
Target: Others
DC41SMe
Cat.No: T10973
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T10018 1-Methyladenine

Others Others
1-Methyladenine is a DNA alkylation product that undergoes damage reversal through oxidative demethylation for repair purposes.

天然产物

1-Methyladenine
Cat.No: T10018
Synonym:
Target: Others
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